Epithalon Paradise Peptides
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Epithalon

Ala-Glu-Asp-Gly. The pineal tetrapeptide behind 30+ years of Russian telomerase and longevity research — now with independent Western replication.

≥99%
Purity
4
Amino Acids
Jul 24
2026 FDA PCAC Review
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Fast shipping across Southeast Asia · Research purposes only
The Science

What is Epithalon?

Epithalon (also spelled Epitalon, and referred to as AEDG after its amino acid code) is a synthetic tetrapeptide — just four amino acids, Ala-Glu-Asp-Gly — developed by Russian scientist Vladimir Khavinson at the St. Petersburg Institute of Bioregulation and Gerontology, starting in the 1980s. It's a synthetic analog of the active component within epithalamin, a polypeptide extract originally isolated from bovine pineal glands.

Epithalon is arguably the flagship compound of an entire Russian research tradition — the "Khavinson bioregulators" — with over 30 years of clinical use in Russian geriatric practice behind it. That's a genuinely long track record, but it comes with an important caveat that deserves stating plainly rather than glossing over: the large-scale human data (a widely cited dataset covering 266 elderly patients, showing 1.6–4.1× fewer deaths over 6–8 years) comes from a single Russian research group, was not blinded or randomized, and has never been independently reproduced at Western clinical trial standards. It's a real, substantial dataset — just not one that's been replicated outside the lab that generated it.

The one piece of genuinely independent validation: a 2025 study by Al-Dulaimi and colleagues, published in Biogerontology, confirmed — in a Western lab, outside Khavinson's own group — that Epithalon extends telomere length in human cell lines via telomerase upregulation or ALT pathway activity. That's a meaningful development: the central telomere claim, first made by Khavinson's lab decades ago, has now been reproduced independently.

4
Amino acids
Ala-Glu-Asp-Gly (AEDG) — one of the smallest peptides in this catalog
30+
Years of research history
Khavinson bioregulator program, St. Petersburg, since the 1980s
2025
Independent replication
Al-Dulaimi et al. confirmed telomere lengthening in a Western lab
Mechanism of Action

How Epithalon works

Epithalon's proposed mechanism has two main strands — one gets far more attention than the other, but both are part of the original research thesis.

🧬
Telomerase Activation
Research reports that Epithalon stimulates hTERT (human telomerase reverse transcriptase) expression — the enzyme responsible for rebuilding telomeres, the protective caps on chromosome ends that shorten with each cell division. Telomere shortening is one of the recognised hallmarks of cellular aging, which is the basis of Epithalon's core longevity claim.
→ Studied telomerase upregulation and telomere maintenance
🌙
Pineal Gland & Melatonin Regulation
Given its pineal-gland origin, Epithalon is studied for restoring age-related decline in melatonin production and normalizing circadian rhythm. Animal studies (Labunets and successors) have shown restoration of pineal melatonin output with Epithalon administration.
→ Studied restoration of circadian and melatonin signalling
🔬
Gene Expression & Epigenetic Modulation
A 2020 Khavinson paper in Molecules described AEDG peptide stimulation of gene expression and neurogenesis through a possible epigenetic mechanism — supporting the broader view that Epithalon's effects may extend beyond telomere biology alone, though this angle is less established than the telomerase work.
→ Broader gene-expression effects under active investigation
Research Areas

What the research actually covers

Epithalon's evidence spans a wide range — from decades-old Russian animal work to a modern 2025 diabetic retinopathy cell study — worth breaking down by what's actually been shown where.

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Telomere Length (independently replicated)
The Al-Dulaimi et al. 2025 Biogerontology study is the most important recent validation — confirming telomere extension via telomerase upregulation or ALT activity in human cell lines, outside Khavinson's own lab. This is the strongest single piece of evidence in Epithalon's research profile.
🐭
Lifespan & Tumor Incidence (animal models)
Anisimov et al. 2003 (Biogerontology) showed Epithalon extended lifespan and reduced spontaneous tumor incidence in SHR mice. A related 2002 paper in the International Journal of Cancer reported reduced mammary tumor incidence in HER-2/neu mice — a preclinical-only oncology signal that shouldn't be over-extrapolated to humans, but is a consistent finding across Khavinson's animal work.
👁️
Retinal Cell Protection (2025, emerging)
A 2025 Italian-Russian collaboration (Gatta, Dovizio, Milillo, Khavinson, Trofimova et al., Stem Cell Reviews and Reports) found Epithalon restored wound healing, reduced reactive oxygen species, and inhibited hyperglycemia-driven epithelial-mesenchymal transition in retinal pigment epithelial cells under diabetic-retinopathy-modeling conditions — a genuinely new research direction beyond the traditional telomere/pineal framing.
⚠️
The Honest Evidence Gap
No Phase 3 randomized controlled trial exists for Epithalon in any indication. The large 266-patient Russian mortality dataset is real but single-lab, non-blinded, and non-randomized. Human replication of most claims is limited to case reports and small open-label studies outside the core telomere work. Weigh the 30-year Russian track record against the thinness of independent Western confirmation.
2026 Regulatory Update

Where Epithalon's regulatory status stands

⚖️
April 22, 2026 — Removed from FDA Category 2
As of April 22, 2026, Epithalon was removed from the FDA's Category 2 bulk drug substance nominations list — the same reorganization wave that affected CJC-1295, MOTS-c, and several other compounds in this catalog. As with those, removal from Category 2 doesn't itself establish a lawful compounding pathway; it opens the door to the formal review that's now scheduled.
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July 24, 2026 — Formal PCAC Review
Epithalon is scheduled for FDA Pharmacy Compounding Advisory Committee review on July 24, 2026, to determine its Section 503A bulk drug substance status. The outcome will determine whether licensed 503A compounding pharmacies may prepare it going forward. This is an active, unresolved process as of mid-2026 — not a settled outcome either way.
🌍
Not Approved by Any Western Regulator
Epithalon has no FDA, EMA, or other Western regulatory approval for any indication. It remains in active clinical use within Russian geriatric practice under the Khavinson bioregulator framework, but that's a different regulatory environment entirely from US or EU frameworks. All Paradise Peptides products are supplied for research purposes only.
Stack Synergies

How Epithalon works with other compounds

Epithalon's own research program has a real, historically documented pairing — but it's worth being upfront that the compound involved isn't currently in this catalog. Here's the honest picture, plus what's practically available today.

📚 The Historical Khavinson Pairing — Epithalon + Thymalin

Worth knowing even though we don't currently stock it: Khavinson's own clinical program consistently shows Epithalon's largest benefits when combined with Thymalin, a separate thymic bioregulator peptide targeting immune function. This is a genuine research-documented combination, not a generic suggestion — but Thymalin is a distinct molecule from anything currently in the Paradise Peptides catalog, so it's mentioned here as context rather than a stack we can currently supply.

🔗 Epithalon + NAD+ — Genomic & Cellular Longevity

The practical pairing available in this catalog today: NAD+ is the coenzyme mitochondria and cells need for energy metabolism and DNA repair machinery, while Epithalon's research focus is telomere maintenance and pineal/circadian regulation. Both sit in the broader cellular-aging research space, addressing different layers of the aging process — genomic stability and circadian signalling from Epithalon, energy metabolism and repair capacity from NAD+ — rather than the same mechanism twice. Worth being clear that this is a complementary research-area pairing rather than a demonstrated pharmacological synergy the way GHRH + GHRP stacks are.

🔬 Epithalon + MOTS-c — Longevity Research Combination

Another reasonable pairing within the catalog: MOTS-c targets mitochondrial energy signalling, Epithalon targets telomere/pineal biology — two different hallmarks-of-aging angles studied alongside each other in the broader longevity research community, though not a combination with dedicated joint trial data of its own.

Research Protocol

Suggested research protocol

1
Reconstitution
Add 2ml bacteriostatic water to a 10mg vial for a concentration of 5mg/ml. Inject BAC water slowly down the side of the vial, never directly onto the powder. Gently swirl; never shake. Use the Paradise Peptides reconstitution calculator for exact syringe marks.
2
Dose range studied
Standard research protocols cite 5–10mg per day, subcutaneously.
3
Cyclical dosing — not continuous
Unlike most other peptides in this catalog, Epithalon is characteristically run in short, defined cycles rather than continuously: 10–20 consecutive days, repeated 2–3 times per year. This cyclical pattern is a consistent feature of the Khavinson research protocols, not an arbitrary choice.
4
Storage
Unreconstituted: −20°C. Reconstituted: +4°C refrigerated, use within 2–3 weeks for best stability. Keep away from light and heat. Do not freeze the reconstituted solution.
FAQ

Frequently asked questions

Is the telomerase claim actually proven?
It's better supported than most longevity-peptide claims, but not "proven" in a strict human clinical sense. A 2025 independent study (Al-Dulaimi et al., outside Khavinson's own lab) confirmed telomere lengthening via telomerase upregulation in human cell lines — genuine, meaningful replication. But no large-scale, randomized, Western human trial has confirmed the same effect in living people. The cell-line result is real; the leap to a human longevity outcome remains unproven.
What about the 266-patient mortality data — is that reliable?
It's a real, substantial dataset — 1.6 to 4.1× fewer deaths over 6–8 years in Khavinson's elderly cohorts — but it comes from a single Russian research group, wasn't blinded or randomized, and has never been independently rerun at Western clinical trial standards. Worth taking seriously as a signal, not as confirmatory proof.
Why is Epithalon dosed in short cycles instead of continuously?
This follows the Khavinson research protocols directly — 10–20 consecutive days, 2–3 times per year, rather than daily year-round use. It's a consistent, deliberate feature of the research program, not a limitation of the compound itself.
What is included in the kit?
For local shipping within the Philippines, every Epithalon order includes a complete research kit: a drawing syringe for reconstitution, insulin syringes for injection, alcohol pads, bacteriostatic water, and secure discreet packaging. For international orders, the kit isn't included by default (some items don't ship well across borders) — the peptide vial ships on its own, and you'll want your own reconstitution supplies on hand. Email us if you're unsure what you'll need.
Can I buy just the peptide vial without the kit?
Yes — if you already have your own supplies, just let us know via email and we'll accommodate you. Email us →
Where does Paradise Peptides ship?
Paradise Peptides is based in Cebu and supplies Epithalon as a research compound across Southeast Asia. Enquiries and orders are handled via email. Shipping is discreet. All products are for research purposes only.
How do I calculate my dose?
Use the free Paradise Peptides reconstitution calculator. Enter your vial size, how much BAC water you added, and your desired dose. The calculator gives you the exact syringe mark — no maths required.
References

Research sources

Al-Dulaimi, et al. Independent replication of Epithalon-induced telomere lengthening via telomerase upregulation and ALT pathway activity in human cell lines. Biogerontology. 2025.
Anisimov VN, et al. Effect of Epithalon on lifespan and spontaneous tumor incidence in SHR mice. Biogerontology. 2003.
Anisimov VN, et al. Reduced mammary tumor incidence with Epithalon in HER-2/neu transgenic mice. International Journal of Cancer. 2002.
Khavinson VK, et al. AEDG peptide stimulation of gene expression and neurogenesis — possible epigenetic mechanism. Molecules. 2020.
Gatta L, Dovizio M, Milillo C, Khavinson VK, Trofimova S, et al. Epitalon effects on retinal pigment epithelial cells under diabetic-retinopathy-modeling conditions. Stem Cell Reviews and Reports. 2025.
Overview of Epitalon — Highly Bioactive Pineal Tetrapeptide with Promising Properties. Comprehensive 40-year research review. International Journal of Molecular Sciences. 2025.
U.S. Food & Drug Administration. Section 503A bulk drug substance list reorganization, April 22, 2026 — Epithalon removed from Category 2 nominations. Pharmacy Compounding Advisory Committee review scheduled July 24, 2026.

The large Khavinson mortality dataset (266 patients) is real but single-lab, non-blinded, and non-randomized — presented here as context, not as confirmatory clinical evidence.

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